Newsletter Volume 40, Number 6, 2025

DMPK 65に掲載予定の論文一覧

[Regular Articles]

Research article

Tyrosine kinase inhibitors, nilotinib and radotinib, suppress both catalytic function and mRNA expression of human cytochrome P450 2J2 and 2C8

Ayaka Kojima, Masayuki Nadai, Hiroshi Yamazaki, Miki Katoh

 

Research article

L-Type amino acid transporter 1-mediated developmental change of cerebral gabapentin distribution across the rat blood-brain barrier

Hiroki Endo, Takeshi Sugouchi, Otaro Kobayashi, Yuma Tega, … Shin-ichi Akanuma

 

Research article

Important role of OATP in the liver disposition of ezetimibe and its consequent glucuronidation metabolite

Ying Su, Xinyi Zhang, Yiguo Jiang, Cheng Wang, Jianqing Ruan

 

Research article

Metabolism of simvastatin by Streptomyces griseolus CYP105A1 and its variants for the production of human simvastatin metabolites

Sachiyo Yoneda, Kaori Yasuda, Bunzo Mikami, Teisuke Takita, … Shinichi Ikushiro

 

Research article

A novel quantitative assessment of formed reactive metabolites by double trapping with [3H]glutathione and [14C]cyanide

Tomoyuki Kawachi, Tatsuki Fukami, Miki Nakajima

 

●各論文のabstractおよび論文内容詳細については,以下のリンクをご覧ください.
Drug Metabolism and Pharmacokinetics | Vol 65, December 2025 | ScienceDirect.com by Elsevier