メインメニュー

第21回年会 ベストポスター賞受賞者とFinalist

第21回日本薬物動態学会年会のベストポスター賞は、エントリーされた87件の演題について予備審査で10件のFinalistに絞られた後、年会時にこの10件の中から3件が選考されました。

演題番号、受賞題名、報告者名、所属は以下の通りです。ベストポスター賞を受賞された皆様、おめでとうございます。 

30PE-23

A NEW METHOD FOR THE PREDICTION OF CLINICAL CYP3A INDUCTION 

Akihisa Kaneko, Motohiro Kato, Nobuo Sekiguchi, Kunihiro Ohta, Atsuko Higashida, Tetsuya Mitsui, and Yoshinori Aso

Chugai Pharmaceutical Co., Ltd.

30PE-32

A New STRATEGY OF HIGH‐SPEED SCREENING AND QUANTITATIVE SAR ANALYSIS TO EVALUATE HUMAN ABC TRANSPORTER ABCG2-DRUG INTERACTIONS 

Hikaru Saito1, Hiroyuki Hirano2, Hiroshi Nakagawa1 and Toshihisa Ishikawa1

1Graduate School of Bioscience and Biotechnology, Tokyo Institute of Technology, 2GS platZ Co. Ltd.,

30PE-61

EVALUATION OF CONDITIONALLY IMMORTALIZED MOUSE BRAIN CAPILLARY ENDOTHELIAL CELLS AS IN VITRO BLOOD-BRAIN BARRIER MODEL BASED ON ABSOLUTE AMOUNT OF TRANSPORTER PROTEINS

Kazunari Yanai2, Junichi Kamiie1,2,3, Yuki Katsukura2, Yumi Sekine2, Satoshi Umezawa1, Ryo Iwase1, Ken Ohmine1,Sumio Ohtsuki1,2,3 and Tetsuya Terasaki1,2,3

1Faculty of Pharmaceutical Sciences and 2Graduate School of Pharmaceutical Sciences, Tohoku University, 3SORST, Japan Science and Technology Agency 

なお、Finalist 10件のうち7件については、下記の通りです。

29PE-08

IMPROVEMENT OF INTESTINAL ABSORPTION BY PEPTIDE-DERIVATION OF NON-ABSORBABLE DRUG VIA PEPTIDE TRANSPORTER PEPT1 

Akihiro Kikuchi1, Michinori Tanaka2, Takahiro Tomoyasu2, Tomoji Maeda1, Ikumi Tamai1

1Department of Molecular Biopharmaceutics, Faculty of Pharmaceutical Sciences, Tokyo University of Science,2Medicinal Chemistry Research Institute, Otsuka Pharmaceutical Co., Ltd.

29PE-16

MOLECULAR IDENTIFICATION AND FUNCTIONAL CHARACTERIZATION OF A pH-SENSITIVE FOLATE TRANSPORTER IN HUMAN INTESTINE

Yasuhiro Nakai1, Katsuhisa Inoue1, Mai Hatakeyama1, Yayoi Hayashi2 and Hiroaki Yuasa1

1Graduate School of Pharmaceutical Sciences, Nagoya City University, 2College of Pharmacy, Kinjo Gakuin University 

29PE-71

RAPID GENOTYPING OF CYP2A6 ALLELES BY FLUORESCENCE RESONANCE ENERGY TRANSFER 

Kazuma Kiyotani1,2, Masaki Fujieda2, Asami Muroi2 and Tetsuya Kamataki1,2

1Faculty of Pharmacy, Takasaki University of Health and Welfare, 2Graduate school of Pharmaceutical Sciences, Hokkaido University 

30PE-59

HUMAN UDP-GLUCURONOSYLTRANSFERASE, UGT1A8, GLUCURONIDATES DIHYDRO-TESTOSTERONE TO A MONOGLUCURONIDE AND FURTHER TO A STRUCTURALLY NOVEL DIGLUCURONIDE

Takahiro Murai, Naozumi Samata, Haruo Iwabuchi and Toshihiko Ikeda

Drug Metabolism and Pharmacokinetics Research Laboratories, Sankyo Co., Ltd., 

30PE-63

INHIBITION OF CHOLINE UPTAKE TRANSPORTER BY GEFITINIB REDUCES PHOSPHATIDYLCHOLINE BIOSYNTHESIS IN PRIMARY CULTURED RAT ALVEOLAR TYPE II CELLS

Masanobu Oyabu1, Naoki Ishiguro1, Toshihiro Sato1, Tomoji Maeda1, Hironobu Minami2 and Ikumi Tamai1

1Faculty of Pharmaceutical Sciences, Tokyo University of Science, 2National Cancer Center Hospital East 

30PE-66

HUMAN UGT1A1, 1A4, 1A6, AND 1A9 INTERACT WITH EACH OTHER TO AFFECT ENZYMATIC ACTIVITIS 

Ryoichi Fujiwara1, Miki Nakajima1, Hiroyuki Yamanaka1, Miki Katoh1, Shin-ichi Ikushiro2, Toshiyuki Sakaki2, and Tsuyoshi Yokoi1

1Graduate School of Medical Science, Kanazawa University, and 2Biotechnology Research Center, Faculty of Engineering, Toyama Prefectural University 

30PE-85

ENERGY-DEPENDENT ORGANIC CATION TRANSPORT SYSTEM IS INVOLVED IN THE BLOOD-BRAIN BARRIER TRANSPORT OF OXYCODONE 

Asami Hattori1, Takashi Okura1, Yusuke Nakazawa1, Rie Ito1, Margareta Hammarlund-Udenaes2, Tetsuya Terasaki3 and Yoshiharu Deguchi1

1School of Pharmaceutical Sciences, Teikyo University, 2Department of Pharmaceutical Biosciences, Uppsala University, 3Graduate School of Pharmaceutical Sciences, Tohoku University